Menthol in biofreeze. Biofreeze: Uses, Side Effects, and Dosage of Menthol-Based Topical Pain Relief

26.08.202308.07.2023 by alexxlab

How does Biofreeze work to relieve pain. What are the potential side effects of using Biofreeze. When should you consult a doctor while using Biofreeze. How should Biofreeze be applied for maximum effectiveness. What precautions should be taken when using Biofreeze.

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Understanding Biofreeze: A Menthol-Based Topical Pain Reliever

Biofreeze is a popular topical pain relief product that contains menthol as its active ingredient. This over-the-counter medication is widely used to alleviate minor aches and pains associated with muscles and joints. Its effectiveness lies in the unique properties of menthol, which acts as a counterirritant on the skin.

How Does Biofreeze Work?

The mechanism of action for Biofreeze is quite fascinating. When applied to the skin, menthol creates a sensation of coolness, which is quickly followed by a warming effect. This alternating temperature sensation helps to distract the brain from pain signals, providing relief to the affected area. This process is known as the gate control theory of pain, where the sensory input from the menthol application essentially “closes the gate” on pain signals reaching the brain.

Common Uses of Biofreeze

Biofreeze is typically used for:

Arthritis pain relief
Backache
Muscle sprains and strains
Joint pain
Minor sports injuries

In some cases, certain brands of menthol-based products may also be used to relieve itching and skin irritation from sunburns, insect bites, or minor scrapes. However, it’s crucial to check the specific product labeling to ensure it’s appropriate for your intended use.

Proper Application and Usage of Biofreeze

To maximize the benefits of Biofreeze while minimizing potential side effects, it’s essential to follow the proper application guidelines.

How to Apply Biofreeze

Here are the steps for applying Biofreeze:

Clean and dry the affected area thoroughly.
Apply a thin layer of the gel, cream, or liquid to the skin.
Gently rub the product into the skin until it’s fully absorbed.
Allow the area to dry completely before covering with clothing.
Wash your hands thoroughly after application unless treating the hands.

Is there a limit to how often Biofreeze can be applied? Yes, it’s recommended to use Biofreeze no more than 3 to 4 times per day on the affected area. Overuse may lead to skin irritation or other adverse effects.

Important Application Tips

Avoid applying Biofreeze to open wounds, cuts, or broken skin.
Do not bandage or tightly wrap the treated area.
Avoid applying heat to the treated area, as this can increase the risk of side effects.
Wait for your skin to cool down before applying Biofreeze after exercise or hot showers.

Potential Side Effects and Precautions

While Biofreeze is generally safe when used as directed, it’s important to be aware of potential side effects and take necessary precautions.

Common Side Effects

The most commonly reported side effects of Biofreeze include:

Redness at the application site
Warmth or mild burning sensation
Skin irritation

These effects are usually mild and temporary. However, if they persist or worsen, it’s advisable to discontinue use and consult a healthcare professional.

Serious Side Effects

While rare, some users may experience more serious side effects. These can include:

Blistering or severe swelling at the application site
Unusual or increased pain in the treated area
Signs of an allergic reaction (rash, itching, swelling, severe dizziness, difficulty breathing)

If you experience any of these serious side effects, stop using the product immediately and seek medical attention.

Precautions and Contraindications

Before using Biofreeze, consider the following precautions:

Inform your doctor or pharmacist about any allergies, especially to menthol.
Disclose your full medical history, as certain conditions may affect the use of this product.
If pregnant or breastfeeding, consult a healthcare provider before use.
Avoid use on children under 12 without medical supervision.

Interactions and Considerations

While Biofreeze is a topical medication, it’s still important to consider potential interactions with other drugs or medical conditions.

Drug Interactions

Can Biofreeze interact with other medications? While topical menthol products like Biofreeze are less likely to interact with systemic medications, it’s always wise to inform your healthcare provider about all products you’re using, including over-the-counter medications and herbal supplements. This helps prevent potential interactions and ensures your overall treatment plan is safe and effective.

Special Considerations

There are certain situations where extra caution is needed when using Biofreeze:

If you have sensitive skin or a history of skin reactions
When using on large areas of the body
If you’re also using other topical medications in the same area
Before undergoing any medical procedures or surgeries

Maximizing the Benefits of Biofreeze

To get the most out of your Biofreeze treatment, consider these tips:

Complementary Therapies

Biofreeze can be used alongside other pain management strategies for enhanced relief:

Gentle stretching exercises
Physical therapy
Rest and proper posture
Cold or heat therapy (but not immediately before or after Biofreeze application)

Lifestyle Modifications

Certain lifestyle changes can complement the pain-relieving effects of Biofreeze:

Maintaining a healthy weight to reduce stress on joints
Regular, low-impact exercise to improve muscle strength and flexibility
Proper ergonomics at work and home to prevent muscle strain
Stress reduction techniques like meditation or deep breathing exercises

When to Seek Medical Advice

While Biofreeze can be effective for many types of minor pain, there are situations where professional medical advice is necessary.

Red Flags

Seek immediate medical attention if you experience:

Severe or persistent pain that doesn’t improve with Biofreeze
Pain accompanied by fever, redness, or swelling
Sudden onset of severe pain
Pain that interferes with daily activities or sleep

Chronic Pain Management

For those dealing with chronic pain conditions, it’s important to work with a healthcare provider to develop a comprehensive treatment plan. Biofreeze can be a part of this plan, but shouldn’t be the sole method of pain management for long-term conditions.

Alternative Menthol-Based Products

While Biofreeze is a popular choice, there are other menthol-based topical pain relievers available on the market. These products may have different concentrations of menthol or additional ingredients that could be more suitable for certain individuals or conditions.

Comparing Options

When considering alternatives to Biofreeze, look at factors such as:

Menthol concentration
Additional active ingredients (e.g., camphor, eucalyptus oil)
Form of application (gel, roll-on, spray)
Price and availability
User reviews and recommendations

Is a higher concentration of menthol always better? Not necessarily. While a higher concentration may provide more intense cooling, it can also increase the risk of skin irritation. It’s often best to start with a lower concentration and increase if needed.

Natural Alternatives

For those preferring natural options, consider:

Peppermint oil (contains natural menthol)
Arnica gel
Capsaicin creams (derived from chili peppers)
Essential oil blends (with proper dilution)

Always conduct a patch test before using any new topical product, especially if you have sensitive skin or allergies.

The Science Behind Menthol’s Pain-Relieving Properties

Understanding the science behind menthol’s effectiveness can help users appreciate how Biofreeze and similar products work to alleviate pain.

Neurological Effects

Menthol’s pain-relieving properties are primarily due to its effects on the nervous system:

Activation of cold-sensitive TRPM8 receptors in skin nerve endings
Desensitization of nociceptors (pain receptors)
Modulation of pain signals in the central nervous system

These neurological effects explain why menthol provides both a cooling sensation and pain relief.

Anti-Inflammatory Properties

Does menthol have anti-inflammatory effects? While primarily known for its analgesic properties, some studies suggest that menthol may also have mild anti-inflammatory effects. This could contribute to its effectiveness in treating muscle and joint pain associated with inflammation.

Circulatory Effects

Menthol’s cooling sensation can lead to vasoconstriction (narrowing of blood vessels) followed by vasodilation (widening of blood vessels). This change in blood flow may contribute to pain relief by:

Reducing inflammation in the affected area
Improving nutrient delivery to tissues
Enhancing removal of waste products from the site of injury

These circulatory effects, combined with the neurological impacts, make menthol a versatile and effective topical pain reliever.

Biofreeze (Menthol) Topical: Uses, Side Effects, Interactions, Pictures, Warnings & Dosing

Uses

Different brands of this product have different uses. Some brands are used to treat minor aches and pains of the muscles/joints (such as arthritis, backache, sprains). Some brands are used to help relieve itching and skin irritation (such as due to sunburn, insect bites, or minor scrapes). Menthol is known as a counterirritant. It works by causing the skin to feel cool and then warm.

How to use Biofreeze (Menthol) 4 % Topical Gel Dermatological Irritants-Counter-Irritant Formulations

If you are using the over-the-counter product to self-treat, read and follow all directions on the product package before using this medication. If you have any questions, consult your pharmacist. If your doctor has prescribed this medication, use it as directed.

This medication is for use on the skin only. Apply to the affected area no more than 3 to 4 times a day. If you are using the cream, gel, or liquid, rub in gently and thoroughly. Some liquid forms of this medication should be shaken before use. Check the manufacturer’s information for specific directions. Let the medicine dry completely before letting anyone else touch the area.

Wash your hands well after applying unless you are using this medication to treat the hands. Avoid getting this medication in your eyes, nose, or mouth. If you do get the medication in those areas, flush with plenty of water.

Do not apply to serious burns or deep wounds. Do not bandage or tightly wrap the affected area. Doing so may increase the risk of side effects. You may cover the area loosely to protect clothing.

Heat can increase the risk of side effects. Do not apply this medication right before, during, or after activities that increase skin temperature (such as bathing, swimming, heavy exercise). Wait until your skin has cooled before applying the medication. Do not use a sunlamp/tanning bed, hot water bottle, or heating pad/device on the treated area.

Check the ingredients on the label even if you have used the product before. The manufacturer may have changed the ingredients. Also, products with similar names may contain different ingredients meant for different purposes. Read the label carefully to make sure you have the right product for you. Ask your pharmacist if you have any questions.

Tell your doctor if your condition lasts for more than 7 days, or if it gets worse, or if it keeps returning. If you think you may have a serious medical problem, get medical help right away.

Side Effects

Redness, warmth, or irritation at the application site may occur. If any of these effects last or get worse, tell your doctor or pharmacist promptly.

If your doctor has directed you to use this medication, remember that your doctor has judged that the benefit to you is greater than the risk of side effects. Many people using this medication do not have serious side effects.

Stop using this medication and tell your doctor right away if you have any serious side effects, including: blistering/swelling at the application site, increased/unusual pain at the application site.

A very serious allergic reaction to this drug is rare. However, get medical help right away if you notice any symptoms of a serious allergic reaction, including: rash, itching/swelling (especially of the face/tongue/throat), severe dizziness, trouble breathing.

This is not a complete list of possible side effects. If you notice other effects not listed above, contact your doctor or pharmacist.

In the US – Call your doctor for medical advice about side effects. You may report side effects to FDA at 1-800-FDA-1088 or at www.fda.gov/medwatch.

In Canada – Call your doctor for medical advice about side effects. You may report side effects to Health Canada at 1-866-234-2345.

Precautions

Before using this product, tell your doctor or pharmacist if you are allergic to menthol; or if you have any other allergies. This product may contain inactive ingredients, which can cause allergic reactions or other problems. Talk to your pharmacist for more details.

Before using this medication, tell your doctor or pharmacist your medical history.

Before having surgery, tell your doctor or dentist about all the products you use (including prescription drugs, nonprescription drugs, and herbal products).

During pregnancy, this medication should be used only when clearly needed. Discuss the risks and benefits with your doctor.

It is unknown if this medication passes into breast milk. Consult your doctor before breast-feeding.

Interactions

Drug interactions may change how your medications work or increase your risk for serious side effects. This document does not contain all possible drug interactions. Keep a list of all the products you use (including prescription/nonprescription drugs and herbal products) and share it with your doctor and pharmacist. Do not start, stop, or change the dosage of any medicines without your doctor’s approval.

Does Biofreeze (Menthol) 4 % Topical Gel Dermatological Irritants-Counter-Irritant Formulations interact with other drugs you are taking?

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Overdose

This medicine may be harmful if swallowed. If someone has overdosed and has serious symptoms such as passing out or trouble breathing, call 911. Otherwise, call a poison control center right away. US residents can call their local poison control center at 1-800-222-1222. Canada residents can call a provincial poison control center.

Keep all regular medical and lab appointments.

If you are using this product on a regular schedule and miss a dose, use it as soon as you remember. If it is near the time of the next dose, skip the missed dose. Use your next dose at the regular time. Do not double the dose to catch up.

Store at room temperature. Different brands of this medication have different storage needs. Check the product package for instructions on how to store your brand, or ask your pharmacist. Keep all medications away from children and pets.

Do not flush medications down the toilet or pour them into a drain unless instructed to do so. Properly discard this product when it is expired or no longer needed. Consult your pharmacist or local waste disposal company.

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Biofreeze (menthol) 4 % topical gel

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Selected from data included with permission and copyrighted by First Databank, Inc. This copyrighted material has been downloaded from a licensed data provider and is not for distribution, except as may be authorized by the applicable terms of use.

CONDITIONS OF USE: The information in this database is intended to supplement, not substitute for, the expertise and judgment of healthcare professionals. The information is not intended to cover all possible uses, directions, precautions, drug interactions or adverse effects, nor should it be construed to indicate that use of a particular drug is safe, appropriate or effective for you or anyone else. A healthcare professional should be consulted before taking any drug, changing any diet or commencing or discontinuing any course of treatment.

Menthol Topical (Biofreeze) – Side Effects, Interactions, Uses, Dosage, Warnings

Brand Names:ActivICE, ActivOn Arthritis, ActivOn Joint and Muscle, Arctic Relief Pain Relieving, Aspercreme Heat Pain Relieving, Asperflex Maximum Strength

Reviewed: January 27, 2022

Menthol is either manmade or made from the extracts of mint oil. Menthol provides a cooling sensation when applied to the skin, which helps relieve pain in the tissues underneath the skin.

Menthol topical (for use on the skin) is used to provide temporary relief of minor arthritis pain, backache, muscles or joint pain, or painful bruises.

There are many brands and forms of menthol available. Not all brands are listed on this leaflet.

Menthol topical may also be used for purposes not listed in this medication guide.

uses

What is Menthol Topical (Biofreeze) used for?

Cough
Pain
Pruritus